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2013
Geurink, P.P., van der Linden, W.A., Mirabella, A.C., Gallastegui, N., de Bruin, G., Blom, A.E.M., Voges, M.J., Mock, E.D., Florea, B. I, van der Marel, G.A., Driessen, C., van der Stelt, M., Groll, M., Overkleeft, H.S., Kisselev, A.F. , Incorporation of Non-natural Amino Acids Improves Cell Permeability and Potency of Specific Inhibitors of Proteasome Trypsin-like Sites, Journal of Medicinal Chemistry, vol. 56, no. 3, pp. 1262-1275. DOI
2012
Kisselev, A.F., van der Linden, W.A., Overkleeft, H.S. , Proteasome Inhibitors: An Expanding Army Attacking a Unique Target, Chemistry & Biology, vol. 19, no. 1, pp. 99-115. DOI
van der Linden, W.A., Li, N., Hoogendoorn, S., Ruben, M., Verdoes, M., Guo, J., Boons, G., van der Marel, G.A., Florea, B. I, Overkleeft, H.S. , Two-step bioorthogonal activity-based proteasome profiling using copper-free click reagents: A comparative study, Bioorganic & Medicinal Chemistry, vol. 20, no. 2, pp. 662-666. DOI
van der Linden, W.A., Willems, L. I, Shabaneh, T.B., Li, N., Ruben, M., Florea, B. I, van der Marel, G.A., Kaiser, M., Kisselev, A.F., Overkleeft, H.S. , Discovery of a potent and highly beta 1 specific proteasome inhibitor from a focused library of urea-containing peptide vinyl sulfones and peptide epoxyketones, Organic & Biomolecular Chemistry, vol. 10, no. 1, pp. 181-194. DOI
Janssen, K.G.H., Li, J., Hoang, H.T., Vulto, P., van den Berg, R.J.B.H.N., Overkleeft, H.S., Eijkel, J.C.T., Tas, N.R., van der Linden, H.J., Hankemeier, T. , Limits of miniaturization: Assessing ITP performance in sub-micron and nanochannels, Lab on a Chip, vol. 12, no. 16, pp. 2888-2893. DOI
2011
Willems, L. I, Van der Linden, W.A., Li, N., Li, K.Y., Liu, N., Hoogendoorn, S., Van der Marel, G.A., Florea, B. I, Overkleeft, H.S. , Bioorthogonal Chemistry: Applications in Activity-Based Protein Profiling, Accounts of Chemical Research, vol. 44, no. 9, pp. 718-729.
2010
Screen, M., Britton, M., Downey, S.L., Verdoes, M., Voges, M.J., Blom, A.E., Guerink, P.P., Risseeuw, M.D., Florea, B. I, van der Linden, W.A., Pletnev, A.A., Overkleeft, H.S., Kisselev, A.F. , The nature of pharmacophore influences active site specificity of proteasome inhibitors, J Biol Chem, vol. 285, pp. 40125-40134. DOI
Verdoes, M., Willems, L. I, van der Linden, W.A., Duivenvoorden, B.A., van der Marel, G.A., Florea, B. I, Kisselev, A.F., Overkleeft, H.S. , A panel of subunit-selective activity-based proteasome probes, Org Biomol Chem, vol. 8, pp. 2719-2727. DOI
van der Linden, W.A., Geurink, P.P., Oskam, C., van der Marel, G.A., Florea, B. I, Overkleeft, H.S. , Proteasome selectivity towards Michael acceptor containing oligopeptide-based inhibitors, Org Biomol Chem, vol. 8, no. 8, pp. 1885-93. DOI
Florea, B. I, Verdoes, M., Li, N., van der Linden, W.A., Geurink, P.P., van den Elst, H., Hofmann, T., de Ru, A., van Veelen, P.A., Tanaka, K., Sasaki, K., Murata, S., den Dulk, H., Brouwer, J., Ossendorp, F.A., Kisselev, A.F., Overkleeft, H.S. , Activity-based profiling reveals reactivity of the murine thymoproteasome-specific subunit beta5t, Chemistry & Biology, vol. 17, pp. 795-801.
2008
Verdoes, M., Florea, B. I, Hillaert, W., Willems, L. I, van der Linden, W.A., Sae-Heng, M., Filippov, D.V., Kisseley, A.F., van der Marel, G.A., Overkleeft, H.S. , Azido-BODIPY acid reveals quantitative Staudinger-Bertozzi ligation in two-step activity-based proteasome profiling, Chembiochem, vol. 9, no. 11, pp. 1735-1738. DOI
2007
Verdoes, M., Florea, B. I, van der Linden, W.A., Renou, D., van den Nieuwendijk, A.M.C.H., van der Marel, G.A., Overkleeft, H.S. , Mixing of peptides and electrophilic traps gives rise to potent, broad-spectrum proteasome inhibitors, Organic & Biomolecular Chemistry, vol. 5, no. 9, pp. 1416-1426. DOI
2006
Verdoes, M., Florea, B. I, Menendez-Benito, V., Maynard, C.J., Witte, M.D., Van der Linden, W.A., Van den Nieuwendijk, A.M.C.H., Hofmann, T., Berkers, C.R., van Leeuwen, F.W.B., Groothuis, T.A., Leeuwenburgh, M.A., Ovaa, H., Neefjes, J.J., Filippov, D.V., van der Marel, G.A., Dantuma, N.P., Overkleeft, H.S. , A fluorescent broad-spectrum proteasome inhibitor for labeling proteasomes in vitro and in vivo, Chemistry & Biology, vol. 13, no. 11, pp. 1217-1226. DOI